Small scale in vitro method to determine a bioequivalent equilibrium solubility range for fasted human intestinal fluid
Volume: 168, Pages: 90 - 96
Published: Nov 1, 2021
Abstract
Drug solubility is a key parameter controlling oral absorption, but intestinal solubility is difficult to assess in vitro. Human intestinal fluid (HIF) aspirates can be applied but they are variable, difficult to obtain and expensive. Simulated intestinal fluids (SIF) are a useful surrogate but multiple recipes are available and the optimum is unknown. A recent study characterised fasted HIF aspirates using a multi-dimensional approach and...
Paper Details
Title
Small scale in vitro method to determine a bioequivalent equilibrium solubility range for fasted human intestinal fluid
Published Date
Nov 1, 2021
Volume
168
Pages
90 - 96
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