Original paper
Intracellular trafficking of new anticancer therapeutics: antibody–drug conjugates
Abstract
: Antibody–drug conjugate (ADC) is a milestone in targeted cancer therapy that comprises of monoclonal antibodies chemically linked to cytotoxic drugs. Internalization of ADC takes place via clathrin-mediated endocytosis, caveolae-mediated endocytosis, and pinocytosis. Conjugation strategies, endocytosis and intracellular trafficking optimization, linkers, and drugs chemistry present a great challenge for researchers to eradicate tumor cells...
Paper Details
Title
Intracellular trafficking of new anticancer therapeutics: antibody–drug conjugates
Published Date
Aug 1, 2017
Volume
Volume 11
Pages
2265 - 2276
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Notes
History