Iron-catalyzed C(5)−H Imidation of Azole with N -Fluorobenzenesulfonimide
Abstract
An iron(II)-catalyzed direct imidation of oxazole and thiazole with N-fluorobenzenesulfonimide (NFSI) through C(5)−H bond cleavage is disclosed, providing C5-imidated azoles in moderate to excellent yields with broad substrate scope. This reaction represents the first iron-catalyzed C−H imidation of arene where NFSI serves as the imidation reagent, and potentially constitutes an efficient access to C5-functionalized azole with great medicinal...
Paper Details
Title
Iron-catalyzed C(5)−H Imidation of Azole with N -Fluorobenzenesulfonimide
Published Date
Oct 18, 2017
Volume
359
Issue
24
Pages
4284 - 4288
Citation AnalysisPro
You’ll need to upgrade your plan to Pro
Looking to understand the true influence of a researcher’s work across journals & affiliations?
- Scinapse’s Top 10 Citation Journals & Affiliations graph reveals the quality and authenticity of citations received by a paper.
- Discover whether citations have been inflated due to self-citations, or if citations include institutional bias.
Notes
History