Iron-catalyzed C(5)−H Imidation of Azole with N -Fluorobenzenesulfonimide

Volume: 359, Issue: 24, Pages: 4284 - 4288
Published: Oct 18, 2017
Abstract
An iron(II)-catalyzed direct imidation of oxazole and thiazole with N-fluorobenzenesulfonimide (NFSI) through C(5)−H bond cleavage is disclosed, providing C5-imidated azoles in moderate to excellent yields with broad substrate scope. This reaction represents the first iron-catalyzed C−H imidation of arene where NFSI serves as the imidation reagent, and potentially constitutes an efficient access to C5-functionalized azole with great medicinal...
Paper Details
Title
Iron-catalyzed C(5)−H Imidation of Azole with N -Fluorobenzenesulfonimide
Published Date
Oct 18, 2017
Volume
359
Issue
24
Pages
4284 - 4288
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