Copper-Catalyzed Direct Amidation of Heterocycles with N-Fluorobenzenesulfonimide
Abstract
A highly efficient amidation reaction of heterocycles with N-fluorobenzenesulfonimide (NFSI) has been developed, presumably proceeding via C-H bond activation. Cuprous iodide was employed as the catalyst, and various α-amidated heterocycle derivatives have been generated in good to excellent yields. This chemistry endowed an economic method of synthesis of valuable amidated heterocycles through a direct C-N bond-coupling...
Paper Details
Title
Copper-Catalyzed Direct Amidation of Heterocycles with N-Fluorobenzenesulfonimide
Published Date
Oct 13, 2014
Journal
Volume
16
Issue
21
Pages
5648 - 5651
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